Author Topic: Styramate analog?  (Read 57 times)

Naphyrone

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Styramate analog?
« on: April 29, 2010, 05:22:32 PM »
I was wondering if anyone had any info on CNS active analogs of Styramate, specifically removing that 2-OH.

Enkidu

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Re: Styramate analog?
« Reply #1 on: April 29, 2010, 08:53:11 PM »
I'm pretty sure it's already centrally active.

Vesp

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Re: Styramate analog?
« Reply #2 on: April 29, 2010, 10:15:00 PM »
Naphyrone, what other bits of information do you have on it? What receptors does it effect, etc?
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Naphyrone

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Re: Styramate analog?
« Reply #3 on: April 30, 2010, 04:17:37 AM »
It is a GABAergic muscle relaxant/sedative/anticonvulsant that effects GABA-a. IUPAC (2-hydroxy-2-phenylethyl) carbamate

Enkidu

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Re: Styramate analog?
« Reply #4 on: April 30, 2010, 07:23:46 AM »
What would be your rational behind an assay of the desoxy version